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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Walter Reed Army Institute Of Research

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMO15-related protein kinase Pfmrk(Plasmodium falciparum)
Walter Reed Army Institute Of Research

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataIC50:  700nMAssay Description:Inhibition of His6x-tagged Plasmodium falciparum Pfmrk expressed in Escherichia coli by microtiter plate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Walter Reed Army Institute Of Research

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Walter Reed Army Institute Of Research

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of human CDK1/cyclin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Homo sapiens (Human))
Walter Reed Army Institute Of Research

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataIC50:  2.09E+5nMAssay Description:Inhibition of human CDK6/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Dalian Institute Of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataEC50:  4.90E+4nMAssay Description:Agonist activity at human FFA1 receptor expressed in CHO-K1 cells assessed as increase in dynamic mass redistribution response by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Dalian Institute Of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50321446(4-methyl-N-(3-(trifluoromethyl)phenyl)benzenesulfo...)
Affinity DataEC50:  2.95E+4nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed