Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 16 hits in this display
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
EC50: 5.70nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium influx by FLIPR assay in presence of 0.1 % BSAMore data for this Ligand-Target Pair
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
EC50: 6.03nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometryMore data for this Ligand-Target Pair
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
EC50: 6.03nMAssay Description:Agonist activity at human GPR40 expressed in Flp-InTM T-RexTM HEK293 cells assessed as stimulation of calcium mobilization in presence of 0.1% BSA by...More data for this Ligand-Target Pair
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
EC50: 14nMAssay Description:Agonist activity at FFA1 receptor (unknown origin) stably expressed in CHO cells assessed as increase in calcium flux by Fluo4-AM based FLIPR assayMore data for this Ligand-Target Pair
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
BDBM50339476(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]-2-fluo...)
EC50: 34.7nMAssay Description:Agonist activity at human GPR40 expressed in Flp-InTM T-RexTM HEK293 cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair