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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Cytochrome P450 2C19
(Homo sapiens (Human))
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
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Affinity Data
IC50: 2.34E+4nM
Assay Description:
Inhibition of CYP2C19 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cytochrome P450 2C9
(Homo sapiens (Human))
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.57E+4nM
Assay Description:
Inhibition of CYP2C9 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucose-dependent insulinotropic receptor
(Rattus norvegicus)
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
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Copy InChI
Affinity Data
EC50: 169nM
Assay Description:
Agonist activity at rat GPR119 by HTRF cAMP assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human))
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
Copy SMILES
Copy InChI
Affinity Data
EC50: 14nM
Assay Description:
Inhibition of human GPR119 activity by homogeneous time resolved fluorescence cyclase (cAMP) assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human))
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
Copy SMILES
Copy InChI
Affinity Data
EC50: 14nM
Assay Description:
Agonist activity at human GPR119 by HTRF cAMP assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucose-dependent insulinotropic receptor
(Rattus norvegicus)
Arena Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50056004
(CHEMBL3326667)
Copy SMILES
Copy InChI
Affinity Data
EC50: 169nM
Assay Description:
Inhibition of rat GPR119 activity by homogeneous time resolved fluorescence cyclase (cAMP) assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI