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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
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Affinity Data
IC50: 30nM
Assay Description:
Binding affinity for human PPAR delta receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Guangdong Pharmaceutical University
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
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Affinity Data
EC50: 325nM
Assay Description:
Agonist activity at human FFA1 receptor expressed in CHO cells by Fluo 4-AM dye based FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor alpha
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.00E+3nM
Assay Description:
Maximum transcriptional activation of human PPAR alpha receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 376nM
Assay Description:
Transactivation of GAL4-fused human PPARdelta LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 90nM
Assay Description:
Maximum transcriptional activation of human PPAR delta receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor gamma
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50127215
(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 7.04E+3nM
Assay Description:
Maximum transcriptional activation of human PPAR gamma receptor
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI