Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL

LigandBDBM50531673(CHEMBL4556462)Copy SMILESCopy InChI

Affinity DataEC50:  1.65E+3nMAssay Description:Transactivation of GAL4-fused human PPARdelta LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL

LigandBDBM50531673(CHEMBL4556462)Copy SMILESCopy InChI

Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FFA1 receptor expressed in CHO cells by Fluo 4-AM dye based FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI