Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of GAL4-fused human PPARalpha LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  102nMAssay Description:Transactivation of GAL4-fused human PPARdelta LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  470nMAssay Description:Agonist activity at Gal4-fused PPARgamma LBD (unknown origin) expressed in HepG2 cells incubated for 18 hrs by dual luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human FFA1 receptor expressed in CHO cells by Fluo 4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50:  67nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells assessed as increase in calcium efflux by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50531655(CHEMBL4579901)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of GAL4-fused human PPARgamma LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed