Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
EC50: >1.00E+4nMAssay Description:Transactivation of GAL4-fused human PPARalpha LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
EC50: 102nMAssay Description:Transactivation of GAL4-fused human PPARdelta LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
EC50: 470nMAssay Description:Agonist activity at Gal4-fused PPARgamma LBD (unknown origin) expressed in HepG2 cells incubated for 18 hrs by dual luciferase reporter assayMore data for this Ligand-Target Pair
EC50: 67nMAssay Description:Agonist activity at FFAR1 (unknown origin) expressed in CHO cells assessed as increase in calcium efflux by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Transactivation of GAL4-fused human PPARgamma LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair