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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 2.90nM
Assay Description:
Inhibition of human FGFR1 by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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Article
PubMed
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Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 4.40nM
Assay Description:
Inhibition of human FGFR3 by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Fibroblast growth factor receptor 2
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 5.20nM
Assay Description:
Inhibition of human FGFR2 by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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In Depth
Details
Article
PubMed
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Target
Fibroblast growth factor receptor 4
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 26nM
Assay Description:
Inhibition of human FGFR4 by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
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Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 210nM
Assay Description:
Inhibition of human KDR by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: 510nM
Assay Description:
Inhibition of human SRC by time-resolved fluorescence or time-resolved fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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In Depth
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Article
PubMed
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Chugai Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50197691
(CHEMBL3891894)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human ERG expressed in CHO cells assessed as reduction in channel currents at -80 mV holding potential by automated whole-cell patch cl...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI