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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Targacept
Curated by
ChEMBL
Ligand
BDBM50161758
(2-(5-chloro-2,3-dihydrobenzo[b]furan-7-ylcarboxami...)
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Affinity Data
Ki: 1nM
Assay Description:
Binding affinity to 5HT3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM50161758
(2-(5-chloro-2,3-dihydrobenzo[b]furan-7-ylcarboxami...)
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Copy InChI
Affinity Data
Ki: 1nM
Assay Description:
Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
5-hydroxytryptamine receptor 4
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM50161758
(2-(5-chloro-2,3-dihydrobenzo[b]furan-7-ylcarboxami...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 280nM
Assay Description:
Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
5-hydroxytryptamine receptor 4
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM50161758
(2-(5-chloro-2,3-dihydrobenzo[b]furan-7-ylcarboxami...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+3nM
Assay Description:
In vitro relaxation of carbachol pre-contracted rat oesophageal TMM.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI