Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 [329-824]
(Homo sapiens (Human))
Novartis
US Patent
Ligand
BDBM355936
(1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0260nM
Assay Description:
The assay employs a short peptide substrate labeled with the single fluorophore PT14 as a fluorescence lifetime probe sensitive to the cleavage state...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1
(Homo sapiens (Human))
Novartis
US Patent
Ligand
BDBM355936
(1-(5-chloro-6-(2H- 1,2,3-triazol-2- yl)pyridin-3-y...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0260nM
Assay Description:
IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI