Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProbable G-protein coupled receptor 142(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  18nMAssay Description:Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed