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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Neuronal acetylcholine receptor subunit alpha-4
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50264883
(3-(2-chlorophenyl)-5-(1-(piperidin-4-yl)-1H-pyrazo...)
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Affinity Data
EC50: 120nM
Assay Description:
Activation of human alpha4beta2 nAChR assessed as potentiation of submaximal response to nicotine induced current
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor subunit alpha-3
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50264883
(3-(2-chlorophenyl)-5-(1-(piperidin-4-yl)-1H-pyrazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Activation of human alpha3beta4 nAChR assessed as potentiation of submaximal response to nicotine induced current
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor subunit alpha-3
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50264883
(3-(2-chlorophenyl)-5-(1-(piperidin-4-yl)-1H-pyrazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Activation of human alpha3beta2 nAChR assessed as potentiation of submaximal response to nicotine induced current
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI