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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Poly(ADP-ribose) glycohydrolase
(Homo sapiens (Human))
Cancer Research Technology
US Patent
Ligand
BDBM370901
(US10239843, Example 8)
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Affinity Data
IC50: 1.33E+3nM
Assay Description:
PARG In vitro assays were conducted in a total volume of 15 ul in a standard 384 well format. 5 ul of Human Full Length PARG (Produced internally by ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Poly(ADP-ribose) glycohydrolase
(Homo sapiens (Human))
Cancer Research Technology
US Patent
Ligand
BDBM370901
(US10239843, Example 8)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.30E+3nM
Assay Description:
Inhibition of PARG in human HeLa cells assessed as induction of MMS-induced PAR chains preincubated for 1 hr followed by MMS addition and measured af...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Poly(ADP-ribose) glycohydrolase
(Homo sapiens (Human))
Cancer Research Technology
US Patent
Ligand
BDBM370901
(US10239843, Example 8)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.30E+3nM
Assay Description:
Inhibition of human full length PARG using Bt-NAD ribosylated PARP1 substrate after 10 mins by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI