Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hit in this display   

TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

US Patent

LigandBDBM542251(US11274090, Example 79 Isomer 2)Copy SMILESCopy InChI

Affinity DataIC50:  97.7nMAssay Description:The full length p300 SPA assay was run following the same protocol as p300 HAT SPA assay, but used 6 nM purified full length p300 (purchased from Act...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
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