Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM60544(BDBM50448674 | US9102669, 46 | US9102669, 63)
BDBM60544(BDBM50448674 | US9102669, 46 | US9102669, 63)
IC50: 23nMT: 2°CAssay Description:The SCD1 enzymatic assay was done in a volume of 50 μL using 10 μg of RLM (prepared as described above) in a 96-well polypropylene plate (e...More data for this Ligand-Target Pair
BDBM60544(BDBM50448674 | US9102669, 46 | US9102669, 63)
BDBM60544(BDBM50448674 | US9102669, 46 | US9102669, 63)
IC50: 25nMAssay Description:Inhibition of SCD1 in human A431 cells assessed as [13C]-palmitic acid conversion to [13C]-palmitoleic acid after 4 hrs by LC/MS analysisMore data for this Ligand-Target Pair
BDBM60544(BDBM50448674 | US9102669, 46 | US9102669, 63)
IC50: 165nMT: 2°CAssay Description:The SCD1 enzymatic assay was done in a volume of 50 μL using 10 μg of RLM (prepared as described above) in a 96-well polypropylene plate (e...More data for this Ligand-Target Pair