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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.20nM
Assay Description:
Binding affinity to BRD4 bromodomain 1 (K57 to E168 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by bromod...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.5nM
Assay Description:
Binding affinity to BRD4 bromodomain 2 (E352 to M457 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by bromo...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.60nM
Assay Description:
Binding affinity to BRD2 bromodomain 1 to 2 (G73 to A560 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by b...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.30nM
Assay Description:
Binding affinity to His-tagged BRD4 bromodomain 1 to 2 (K57 to K550 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain testis-specific protein
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5.90nM
Assay Description:
Binding affinity to BRDT bromodomain 1 to 2 (N21to P380 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by br...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
Ki: 17nM
Assay Description:
Binding affinity to BRD3 bromodomain 1 to 2 (P24 to P416 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by b...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Abbvie
Curated by
ChEMBL
Ligand
BDBM50457495
(CHEMBL4215988)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.5nM
Assay Description:
Binding affinity to BRD4 in human H1299 cells stably expressing E2 and HPV16-LCR luciferase reporter incubated for 24 hrs by Bright-Glo luciferase re...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI