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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataKi:  99nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  44nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  141nMAssay Description:Agonist activity at GPR119 in human HEK293 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400775(CHEMBL2204982)
Affinity DataEC50:  63nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed