Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetHistone deacetylase 8(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094216(CHEMBL3585983)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094216(CHEMBL3585983)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094216(CHEMBL3585983)
Affinity DataIC50:  8.25E+3nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed