Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProlyl endopeptidase(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50557410(CHEMBL4751873)Copy SMILESCopy InChI

Affinity DataIC50:  9nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50557410(CHEMBL4751873)Copy SMILESCopy InChI

Affinity DataIC50:  50nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50557410(CHEMBL4751873)Copy SMILESCopy InChI

Affinity DataIC50:  200nMAssay Description:Inhibition of DPP4 (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI