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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
TRAF2 and NCK-interacting protein kinase
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 26nM
Assay Description:
Inhibition of human recombinant TNIK (1 to 367 residues) using RLGRDKYKTLRQIRQ as substrate in presence of ATP incubated for 40 mins by radiometric b...
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Target Info
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Target
Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 30nM
Assay Description:
Inhibition of human recombinant FLT4 (800 to end residues) using GGEEEEYFELVKKKK as substrate in presence of ATP incubated for 40 mins by radiometric...
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Target Info
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 191nM
Assay Description:
Inhibition of human recombinant FLT1 (783 to end residues) using KKKSPGEYVNIEFG as substrate in presence of ATP incubated for 40 mins by radiometric ...
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Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 441nM
Assay Description:
Inhibition of full length human recombinant DRAK1 using KKLNRTLSFAEPG as substrate in presence of ATP incubated for 40 mins by radiometric based scin...
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Target
Aurora kinase A
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 517nM
Assay Description:
Inhibition of full length human recombinant AURORA-A using LRRASLG as substrate in presence of ATP incubated for 40 mins by radiometric based scintil...
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Target Info
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Target
Hexokinase-4
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 3.66E+3nM
Assay Description:
Inhibition of human recombinant GCK (1 to 473 residues) using myelin basic protein as substrate in presence of ATP incubated for 40 mins by radiometr...
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Target Info
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Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
Sichuan University
Curated by
ChEMBL
Ligand
BDBM50602947
(CHEMBL5181357)
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Affinity Data
IC50: 4.55E+3nM
Assay Description:
Inhibition of human MLK3 in presence of ATP by radiometric assay
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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antibodypedia
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