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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetTRAF2 and NCK-interacting protein kinase(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant TNIK (1 to 367 residues) using RLGRDKYKTLRQIRQ as substrate in presence of ATP incubated for 40 mins by radiometric b...More data for this Ligand-Target Pair
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TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant FLT4 (800 to end residues) using GGEEEEYFELVKKKK as substrate in presence of ATP incubated for 40 mins by radiometric...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  191nMAssay Description:Inhibition of human recombinant FLT1 (783 to end residues) using KKKSPGEYVNIEFG as substrate in presence of ATP incubated for 40 mins by radiometric ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  441nMAssay Description:Inhibition of full length human recombinant DRAK1 using KKLNRTLSFAEPG as substrate in presence of ATP incubated for 40 mins by radiometric based scin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase A(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  517nMAssay Description:Inhibition of full length human recombinant AURORA-A using LRRASLG as substrate in presence of ATP incubated for 40 mins by radiometric based scintil...More data for this Ligand-Target Pair
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TargetHexokinase-4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  3.66E+3nMAssay Description:Inhibition of human recombinant GCK (1 to 473 residues) using myelin basic protein as substrate in presence of ATP incubated for 40 mins by radiometr...More data for this Ligand-Target Pair
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TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50602947(CHEMBL5181357)
Affinity DataIC50:  4.55E+3nMAssay Description:Inhibition of human MLK3 in presence of ATP by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails PubMed