Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetProthrombin(Bos taurus (Bovine))
University Of Bari &Quot;Aldo Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50442072(CHEMBL2441058)
Affinity DataKi:  211nMAssay Description:Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari &Quot;Aldo Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50442072(CHEMBL2441058)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Bari &Quot;Aldo Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50442072(CHEMBL2441058)
Affinity DataKi:  6.87E+4nMAssay Description:Inhibition of human neutrophil leukocyte elastase using N-(methoxysuccinyl)-Ala-Ala-Pro-Val-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
University Of Bari &Quot;Aldo Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50442072(CHEMBL2441058)
Affinity DataKi:  7.16E+4nMAssay Description:Inhibition of bovine alpha-chymotrypsin using N-succinyl-Ala-Ala-Pro-Phe-p-NA as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
University Of Bari &Quot;Aldo Moro&Quot

Curated by ChEMBL
LigandPNGBDBM50442072(CHEMBL2441058)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human recombinant factor 7a using spectrozyme as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed