Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target26S proteasome non-ATPase regulatory subunit 11(Human)
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50519236(CHEMBL3586646)Copy SMILESCopy InChI

Affinity DataKd:  8.53E+3nMAssay Description:Binding affinity to biotinylated recombinant Rpn6 (unknown origin) assessed as dissociation constant by biolayer interferometry analysisMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI

TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL

LigandBDBM50519236(CHEMBL3586646)Copy SMILESCopy InChI

Affinity DataKd: >1.20E+5nMAssay Description:Binding affinity to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance ...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI