Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279331((1R,5S)-3-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-1,2,3,...)
Affinity DataKi:  670nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279331((1R,5S)-3-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-1,2,3,...)
Affinity DataKi:  965nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279331((1R,5S)-3-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-1,2,3,...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed