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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Beta-adrenergic receptor kinase 1
(Bos taurus)
University of Michigan
Curated by
ChEMBL
Ligand
BDBM50260149
(CHEMBL4074476)
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Affinity Data
IC50: 3.02E+3nM
Assay Description:
Inhibition of bovine GRK2 S670A mutant after 5 mins in presence of ATP by phosphorimaging assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
G protein-coupled receptor kinase 5
(Bos taurus)
University of Michigan
Curated by
ChEMBL
Ligand
BDBM50260149
(CHEMBL4074476)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of bovine GRK5 after 5 mins after 5 mins in presence of ATP by phosphorimaging assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Rhodopsin kinase GRK1
(Bos taurus)
University of Michigan
Curated by
ChEMBL
Ligand
BDBM50260149
(CHEMBL4074476)
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Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Binding affinity of compound towards dopamine transporter determined using [3H]WIN-35 428 as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI