Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-adrenergic receptor kinase 1(Bos taurus)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50260133(CHEMBL4077197)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of bovine GRK2 S670A mutant after 5 mins in presence of ATP by phosphorimaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-coupled receptor kinase 5(Bos taurus)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50260133(CHEMBL4077197)
Affinity DataIC50:  7.63E+4nMAssay Description:Binding affinity towards norepinephrine transporter determined using [3H]nisoxetine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhodopsin kinase GRK1(Bos taurus)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50260133(CHEMBL4077197)
Affinity DataIC50: >1.00E+5nMAssay Description:Ki value against bovine alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed