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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Neutral amino acid transporter B(0)
(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by
ChEMBL
Ligand
BDBM50088534
(CHEMBL3576929 | US10189805, Compound 5)
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Affinity Data
IC50: 3.12E+5nM
Assay Description:
Inhibition of ASCT2-mediated [3H]glutamine uptake in HEK293 cells after 15 mins by Live-cell glutamine uptake assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Neutral amino acid transporter B(0)
(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by
ChEMBL
Ligand
BDBM50088534
(CHEMBL3576929 | US10189805, Compound 5)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.12E+5nM
Assay Description:
The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Neutral amino acid transporter B(0)
(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by
ChEMBL
Ligand
BDBM50088534
(CHEMBL3576929 | US10189805, Compound 5)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.12E+5nM
Assay Description:
Inhibition of ASCT2 (unknown origin)-mediated glutamine transport
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI