Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50088534(CHEMBL3576929 | US10189805, Compound 5)
Affinity DataIC50:  3.12E+5nMAssay Description:Inhibition of ASCT2-mediated [3H]glutamine uptake in HEK293 cells after 15 mins by Live-cell glutamine uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50088534(CHEMBL3576929 | US10189805, Compound 5)
Affinity DataIC50:  3.12E+5nMAssay Description:The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50088534(CHEMBL3576929 | US10189805, Compound 5)
Affinity DataIC50:  3.12E+5nMAssay Description:Inhibition of ASCT2 (unknown origin)-mediated glutamine transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed