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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histamine H4 receptor
(Rattus norvegicus (rat))
Abbott Laboratories
Ligand
BDBM26396
(2,4-diamino-5,6-disubstituted pyrimidine, 10 | 6-[...)
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Affinity Data
Ki: 3.80nM ΔG°: -48.1kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Abbott Laboratories
Ligand
BDBM26396
(2,4-diamino-5,6-disubstituted pyrimidine, 10 | 6-[...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.70nM ΔG°: -47.5kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Abbott Laboratories
Ligand
BDBM26396
(2,4-diamino-5,6-disubstituted pyrimidine, 10 | 6-[...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5nM
Assay Description:
Displacement of [3H]histamine from human H4 receptor expressed in HEK cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI