Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 7.20nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 7.20nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 9nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 9nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 10nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 49nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 49nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 81nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 81nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 1.20E+3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 1.20E+3nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 7.20E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 9.00E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 1.00E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 4.90E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 8.10E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514532(US11096924, DASH-inhibitors 3102 A | US11583516, C...)
IC50: 1.20E+6nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair