Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed