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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCoagulation factor X(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM50176243(2-(1H-imidazol-4-yl)-1H-benzoimidazole-5-carboxami...)
Affinity DataKi:  30nMAssay Description:Binding affinity to FXa in presence of Zn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM50176243(2-(1H-imidazol-4-yl)-1H-benzoimidazole-5-carboxami...)
Affinity DataKi:  900nMAssay Description:Binding affinity to FVIIa in presence of Zn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM50176243(2-(1H-imidazol-4-yl)-1H-benzoimidazole-5-carboxami...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to thrombin in presence of Zn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM50176243(2-(1H-imidazol-4-yl)-1H-benzoimidazole-5-carboxami...)
Affinity DataKi:  3.80E+4nMAssay Description:Binding affinity to FXa in absence of Zn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM50176243(2-(1H-imidazol-4-yl)-1H-benzoimidazole-5-carboxami...)
Affinity DataKi:  3.70E+5nMAssay Description:Binding affinity to FVIIa in absence of Zn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 3(Homo sapiens (Human))
The Josip Juraj Strossmayer University

LigandPNGBDBM85260(Benzimidazole derivative, 1)
Affinity DataIC50:  5.30E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed