Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPlasma kallikrein(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL

LigandBDBM14917(2-[3-(5-carbamimidoyl-1H-1,3-benzodiazol-2-yl)-5-(...)Copy SMILESCopy InChI

Affinity DataKi:  3nMAssay Description:Binding affinity to plasma kallikreinMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetCoagulation factor VII(Homo sapiens (Human))
Celera

LigandBDBM14917(2-[3-(5-carbamimidoyl-1H-1,3-benzodiazol-2-yl)-5-(...)Copy SMILESCopy InChI

Affinity DataKi:  66nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI