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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCoagulation factor VII(Homo sapiens (Human))
Celera

LigandPNGBDBM14864(5-azaindole analog 2 | {[3-(2-hydroxy-3-{1H-pyrrol...)
Affinity DataKi:  800nM ΔG°:  -34.4kJ/molepH: 7.4 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Celera

LigandPNGBDBM14864(5-azaindole analog 2 | {[3-(2-hydroxy-3-{1H-pyrrol...)
Affinity DataKi:  4.65E+4nM ΔG°:  -24.5kJ/molepH: 7.4 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Celera

LigandPNGBDBM14864(5-azaindole analog 2 | {[3-(2-hydroxy-3-{1H-pyrrol...)
Affinity DataKi:  7.15E+4nM ΔG°:  -23.4kJ/molepH: 7.4 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Celera

LigandPNGBDBM14864(5-azaindole analog 2 | {[3-(2-hydroxy-3-{1H-pyrrol...)
Affinity DataKi:  1.25E+5nM ΔG°:  -22.1kJ/molepH: 7.4 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed