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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  10nMAssay Description:Inhibition of Plasmodium falciparum LAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  36nMAssay Description:Inhibition of porcine APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  36nMAssay Description:Inhibition of APN in porcine kidney using L-leucine p-nitroanilide as substrate preincubated for 60 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Sus scrofa)
Wroc?Aw University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  6.47E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed