Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi:  2.51E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi: <1.00E+5nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataEC50:  2.82E+3nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataEC50:  8.51E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed