Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
IC50: 37.1nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
IC50: 37.1nMpH: 4.2Assay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
IC50: 1.28E+6nMpH: 3.5Assay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
BDBM171463(US9085576, 97 | US9085576, 99 | US9611261, Example...)
IC50: 1.28E+6nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair