Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM314810(N-(6- 9((1RS),(5S,R),(6R,S))- 3-amino-5- (difluoro...)
BDBM171700(US9085576, 330 | US9085576, 331)
BDBM171700(US9085576, 330 | US9085576, 331)
IC50: 2.67E+4nMpH: 4.2Assay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
BDBM314810(N-(6- 9((1RS),(5S,R),(6R,S))- 3-amino-5- (difluoro...)
BDBM171700(US9085576, 330 | US9085576, 331)
BDBM171700(US9085576, 330 | US9085576, 331)
IC50: 1.51E+6nMpH: 3.5Assay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair