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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-secretase 2(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM338846((rac)-N-{3-[4-amino-6-(fluoromethyl)-6,7-dihydro[1...)
Affinity DataIC50:  501nMAssay Description:This assay is a Fluorescence Resonance Energy Transfer Assay (FRET) based assay. The substrate for this assay contains the ¿Swedish¿ Lys-Met/Asn-Leu ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM338846((rac)-N-{3-[4-amino-6-(fluoromethyl)-6,7-dihydro[1...)
Affinity DataIC50:  759nMAssay Description:This assay is a Fluorescence Resonance Energy Transfer Assay (FRET) based assay. The substrate for this assay is an APP derived 13 amino acids peptid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM338846((rac)-N-{3-[4-amino-6-(fluoromethyl)-6,7-dihydro[1...)
Affinity DataIC50:  1.00E+9nMAssay Description:This assay is a Fluorescence Resonance Energy Transfer Assay (FRET) based assay. The substrate for this assay is an APP derived 13 amino acids peptid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent