Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM23990(3-amino-1,2,3,4-tetrahydroquinolin-2-one hydrochlo...)
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrsMore data for this Ligand-Target Pair
BDBM23990(3-amino-1,2,3,4-tetrahydroquinolin-2-one hydrochlo...)
BDBM23990(3-amino-1,2,3,4-tetrahydroquinolin-2-one hydrochlo...)
BDBM23990(3-amino-1,2,3,4-tetrahydroquinolin-2-one hydrochlo...)
IC50: >1.00E+6nMAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair