Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: 2.65E+3nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of lysine gingipain were measured in a fluorogenic assay similar to thos...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of cathepsins B, H, K, L, and S were measured in similar assays. Boc-Leu...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of cathepsins B, H, K, L, and S were measured in similar assays. Boc-Leu...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of cathepsins B, H, K, L, and S were measured in similar assays. Boc-Leu...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of lysine gingipain were measured in a fluorogenic assay similar to thos...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of lysine gingipain were measured in a fluorogenic assay similar to thos...More data for this Ligand-Target Pair
BDBM453293(US10730826, Compound 4a | US11325884, Compound 4a)
IC50: >1.00E+5nMAssay Description:The capacities of compounds of the present invention to inhibit the activity of lysine gingipain were measured in a fluorogenic assay similar to thos...More data for this Ligand-Target Pair