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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistone acetyltransferase p300(Homo sapiens (Human))
Avera Institute For Human Genetics

Curated by ChEMBL
LigandPNGBDBM50511824(CHEMBL4451922)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged p300 HAT domain (1195 to 1673 residues) expressed in Escherichia coli BL21 codon plus cells using Histone ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50511824(CHEMBL4451922)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50511824(CHEMBL4451922)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition Dengue serotype-2 NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50511824(CHEMBL4451922)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed