Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCoagulation factor VII(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215435(CHEMBL243108 | N-{[4-(N-aminocarbamimidoyl)phenyl]...)
Affinity DataIC50:  7.02E+3nMAssay Description:Inhibition of factor 7aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215435(CHEMBL243108 | N-{[4-(N-aminocarbamimidoyl)phenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215435(CHEMBL243108 | N-{[4-(N-aminocarbamimidoyl)phenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of factor 2aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed