Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50256515(CHEMBL475776 | N-(5-phenyl-1,3,4-thiadiazol-2-yl)s...)
Ki: 870nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256515(CHEMBL475776 | N-(5-phenyl-1,3,4-thiadiazol-2-yl)s...)
Ki: 1.66E+3nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 1 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256515(CHEMBL475776 | N-(5-phenyl-1,3,4-thiadiazol-2-yl)s...)
Ki: 5.54E+3nMAssay Description:Inhibition of truncated human cloned membrane-associated carbonic anhydrase 4 preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256515(CHEMBL475776 | N-(5-phenyl-1,3,4-thiadiazol-2-yl)s...)
Ki: 7.50E+3nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5B preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256515(CHEMBL475776 | N-(5-phenyl-1,3,4-thiadiazol-2-yl)s...)
Ki: 9.20E+3nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5A pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair