Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
Carbonic anhydrase 2(Homo sapiens (Human))University of Agricultural Sciences and Veterinary Medicine
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
Carbonic anhydrase 9(Homo sapiens (Human))University of Agricultural Sciences and Veterinary Medicine
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
Carbonic anhydrase 4(Bos taurus (bovine))University of Agricultural Sciences and Veterinary Medicine
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
Ki: 3.19E+3nM ΔG°: -31.4kJ/molepH: 8.3 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
Carbonic anhydrase 1(Homo sapiens (Human))University of Agricultural Sciences and Veterinary Medicine
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
BDBM11606(β-CA inhibitor, 5 | 4-Amino-5-bromo-3-fluorob...)
Ki: 4.31E+3nM ΔG°: -30.6kJ/molepH: 8.3 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair