Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278224(CHEMBL4162854)
Affinity DataIC50:  200nMAssay Description:Compound was tested for Antagonistic activity against denuded rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278267(CHEMBL4161404)
Affinity DataIC50:  200nMAssay Description:Compound was tested for Antagonistic activity against denuded rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278224(CHEMBL4162854)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human HDAC1 using p53 (379 to 382 residues) derived fluorogenic peptide RHKKAcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278224(CHEMBL4162854)
Affinity DataIC50:  2.10E+3nMAssay Description:H3 -antagonist potency determined in electrically stimulated guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278267(CHEMBL4161404)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human HDAC2 using p53 (379 to 382 residues) derived fluorogenic peptide RHKKAcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278267(CHEMBL4161404)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human HDAC1 using p53 (379 to 382 residues) derived fluorogenic peptide RHKKAcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed