Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278223(CHEMBL4173137)
Affinity DataIC50:  800nMAssay Description:Compound was tested for its potency against 5-hydroxytryptamine 1A receptor in rat frontal cortex membranes (experiment 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278223(CHEMBL4173137)
Affinity DataIC50:  800nMAssay Description:Inhibition of full length human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 (395 to 489 residues) co-expressed in baculovirus infected sf...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278223(CHEMBL4173137)
Affinity DataIC50:  1.10E+3nMAssay Description:H3 -antagonist potency determined in electrically stimulated guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50278223(CHEMBL4173137)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human HDAC1 using p53 (379 to 382 residues) derived fluorogenic peptide RHKKAcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed