Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetP2Y purinoceptor 1(Meleagris gallopavo)
National Institute Of Diabetes

Curated by ChEMBL

LigandBDBM50118226(CHEMBL337062 | PAPET-ATP)Copy SMILESCopy InChI

Affinity DataEC50:  1.5nMAssay Description:Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of turkey erythrocytesMore data for this Ligand-Target Pair

Target InfoMMDBKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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TargetP2X purinoceptor 4(RAT)
National Institute Of Diabetes

Curated by ChEMBL

LigandBDBM50118226(CHEMBL337062 | PAPET-ATP)Copy SMILESCopy InChI

Affinity DataEC50:  1.50E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetP2X purinoceptor 2(RAT)
National Institute Of Diabetes

Curated by ChEMBL

LigandBDBM50118226(CHEMBL337062 | PAPET-ATP)Copy SMILESCopy InChI

Affinity DataEC50:  1.00E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X4) at 30 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetP2X purinoceptor 1(RAT)
National Institute Of Diabetes

Curated by ChEMBL

LigandBDBM50118226(CHEMBL337062 | PAPET-ATP)Copy SMILESCopy InChI

Affinity DataEC50:  98nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 1 (P2X1) at 1 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetP2X purinoceptor 3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL

LigandBDBM50118226(CHEMBL337062 | PAPET-ATP)Copy SMILESCopy InChI

Affinity DataEC50:  17nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 3 (P2X3) at 10 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI