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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180749(2-(thiazol-4-yl)-1H-benzo[d]imidazol-5-amine | 5-a...)
Affinity DataIC50:  3.39E+3nMAssay Description:Inhibition of Co2+ loaded MetAP expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Universit£T Heidelberg

Curated by ChEMBL
LigandPNGBDBM50180749(2-(thiazol-4-yl)-1H-benzo[d]imidazol-5-amine | 5-a...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed