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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50384019
(CHEMBL2032285 | CHEMBL2079397)
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Affinity Data
IC50: 3.60nM
Assay Description:
Inhibition of recombinant FLT3 by time resolved-fluorescence resonance energy transfer analysis
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
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Article
PubMed
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50384019
(CHEMBL2032285 | CHEMBL2079397)
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Affinity Data
IC50: 14nM
Assay Description:
Inhibition of recombinant c-Met by time resolved-fluorescence resonance energy transfer analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50384019
(CHEMBL2032285 | CHEMBL2079397)
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Affinity Data
IC50: 1.94E+3nM
Assay Description:
Inhibition of GRK-5 (unknown origin) preincubated with enzyme for 10 mins before adding peptide substrate and ATP measured after 1 hr by LANCE-TR-FRE...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Beta-adrenergic receptor kinase 1
(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50384019
(CHEMBL2032285 | CHEMBL2079397)
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Affinity Data
IC50: 6.20E+3nM
Assay Description:
Inhibition of GRK-2 (unknown origin) preincubated with enzyme for 10 mins before adding peptide substrate and ATP measured after 1 hr by LANCE-TR-FRE...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI