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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282489(1-Naphthylamine | CHEBI:50450 | CHEMBL57394 | Naph...)
Affinity DataIC50:  1.81E+5nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50282489(1-Naphthylamine | CHEBI:50450 | CHEMBL57394 | Naph...)
Affinity DataKd:  1.20E+6nMAssay Description:Binding affinity to human recombinant His-tagged Keap1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissoc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed