Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 27 hits in this display
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
IC50: 250nMAssay Description:Inhibition of N-terminal GST-tagged human BRAF/MEK1/RAF1 Y340D/Y341D double mutant measured after 2 hrs in presence of ATP by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)
BDBM50072147((2Z,3Z)-2,3-bis(amino(2-aminophenylthio)methylene)...)