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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMpH: 7.0 T: 2°CAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  14.5nMAssay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  128nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent